Guasch L., Zakharov A., Tarasova O., Poroikov V.V, Liao C., Nicklaus M.C. Novel HIV-1 integrase inhibitor development by virtual screening based on QSAR models // Curr. Top. Med. Chem.- 2015.- Vol. 16, № 4.- Р. 441-448.
Kramer C., Kalliokoski T., Gedeck P., Vulpetti A. The experimental uncertainty of heterogeneous public K(i) data // J. Med. Chem.- 2012.- Vol. 55, № 11.- Р. 5165-5173.
Tarasova O., Urusova A., Filimonov D., Nicklaus M.C., Zakharov A.V., Poroikov V.V. QSAR Modeling Using Large-Scale Databases: Case Study for HIV-1 Reverse Transcriptase Inhibitors // J. Chem. Inf. Model.- 2015.- Vol. 55, № 7.- Р. 1388-1399.
Filimonov D., Zakharov A., Lagunin A., Poroikov V.V.QNA based «Star Track» QSAR approach // SAR and QSAR Environ. Res.- 2009.- Vol. 20, № 7-8.- Р. 679-709.
Zakharov A., Peach M., Sitzmann M., Nicklaus M.C. A new approach to radial basis function approximation and its application to QSAR // J. Chem. Inf. Model.- 2014.- Vol. 54, № 3.- Р. 713-719.
Berthold M., Cebron N., Dill F., Gabriel T., Kötter T., Meinl T., Ohl P., Sieb C., Thiel K., Wieswedel K. The Konstanz Information Miner. In: Studies in Classification, Data Analysis, and Knowledge Organization. Springer, Heidelberg, 2007.
Kelly T., Proudfoot J., McNeil D., Patel U., David E., Hargrave K., Grob P., Cardozo M., Agarwal A., Adams J. Novel non-nucleoside inhibitors of human immunodeficiency virus type 1 reverse transcriptase. 6.2-Indol-3-yl- and 2-azaindol-3-yl-dipyridodiazepinones // J. Med. Chem.- 1997.- Vol. 40, № 15.- Р. 2430-2433.
Mai A., Sbardella G., Artico M., Massa S., Novellino E., Greco G., Lavecchia А. Structure-based design, synthesis, and biological evaluation of conformationally restricted novel 2-alkylthio-6-[1-(2,6-difluorophenyl)alkyl]-3,4-dihydro-5-alkylpyrimidin-4(3H)-ones as non-nucleoside inhibitors of HIV-1 reverse transcriptase // J. Med. Chem.- 2001.- Vol. 44, № 16.- Р. 2544-2554.
Wyatt P., Bethell R., Cammack N., Charon D., Dodic N., Dumaitre B., Evans D., Green D., Hopewell P., Humber D., Lamont R., Orr D., Plested S., Ryan M., Sollis S., Storer R., Weingarten G. Benzophenone derivatives: a novel series of potent and selective inhibitors of human immunodeficiency virus type 1 reverse transcriptase // J. Med. Chem.- 1995.- Vol. 38, № 10.- Р. 1657-1665.
O’Meara J., Yoakim C., Bonneau P., Bos M., Cordingley M., Deziel R., Doyon L. Novel 8-substituted dipyridodiazepinone inhibitors with a broad-spectrum of activity against HIV-1 strains resistant to non-nucleoside reverse transcriptase inhibitors // J. Med. Chem.- 2005.- Vol. 48, № 17.- Р. 5580-5588.
Orchard S., Al-Lazikani B., Bryant S., Clark D., Calder E. Minimum information about a bioactive entity (MIABE) // Nat. Rev. Drug. Discov.- 2011.- Vol. 10, № 9.- Р. 661-669